A new synthesis of amino substituted azolo[1,3,5]triazines via reaction of N1,N1-dimethyl-N2-azolylformamidines with cyanamide
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Open access
Authors
Kalinin, D.
Kalinina, S.
Dolzhenko, Anton
Date
2013Type
Journal Article
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Kalinin, Dimitrii V. and Kalinina, Svetlana A. and Dolzhenko, Anton V. 2013. A new synthesis of amino substituted azolo[1,3,5]triazines via reaction of N1,N1-dimethyl-N2-azolylformamidines with cyanamide. Heterocycles. 87 (1): pp. 147-154.
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Heterocycles
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Publisher can be found at: http://www.heterocycles.jp/newlibrary/libraries/prepress
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Abstract
The amino substituted triazine ring was annelated to aminoazoles using a new effective synthetic procedure. The method of preparation involved initial formation of azolylformamidines in the reaction of aminoazoles with N,N-dimethylformamide dimethyl acetal followed by the triazine ring closure with cyanamide affording therefore fused aminotriazines.
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